Acetylcholinesterase function
Cholinesterase is an enzyme that breaks down acetylcholine into choline and acetic acid, a reaction necessary to allow a cholinergic neuron to return to its resting state after activation.
There are two types of
cholinesterases:
Acetylcholinesterase, also known as RBC cholinesterase, erythrocyte
cholinesterase, or acetylcholine acetylhydrolase, found mostly in the blood and
neural synapses.
Pseudocholinesterase, also known as plasma cholinesterase, butyrylcholinesterase,
or acylcholine acylhydrolase, found mostly in the liver.
Acetylcholinesterase hydrolyses acetylcholine more quickly; Pseudocholinesterase
hydrolyses butyrylcholine more quickly.
Many plants have
acetylcholinesterase inhibitor activity, here is one example"
In vitro acetylcholinesterase inhibitory activity of the essential oil
from Acorus calamus and its main constituents.
Planta Med. 2007; Mukherjee PK, Kumar V, Mal M. School of
Natural Product Studies, Department of Pharmaceutical Technology, Jadavpur
University, Kolkata, India.
The in vitro acetylcholinesterase inhibitory potential of the hydroalcoholic
extract and of the essential oil from Acorus calamus rhizomes and that of its
major constituents were evaluated. Analysis of the oil revealed that the major
constituents were beta-asarone (79%) and alpha-asarone (8%). The experimental
observations revealed that the Acorus calamus essential oil and its constituents
have significant acetylcholinesterase inhibitory potential. beta-Asarone, the
major phytoconstituent present in the essential oil, showed the maximum
inhibitory potential.
Galantamine is a cholinesterase inhibitor substance available without a prescription.